Compile Data Set for Download or QSAR
Report error Found 101 Enz. Inhib. hit(s) with all data for entry = 50002663
TargetCathepsin K(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461260(CHEMBL4228926)
Affinity DataIC50: 0.110nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461249(CHEMBL1215628)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461249(CHEMBL1215628)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461249(CHEMBL1215628)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461256(CHEMBL4228143)
Affinity DataIC50: 1nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461256(CHEMBL4228143)
Affinity DataIC50: 1nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461260(CHEMBL4228926)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461265(CHEMBL4226307)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461248(CHEMBL4227295)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461271(CHEMBL4224764)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461272(CHEMBL4227031)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461269(CHEMBL4227166)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461270(CHEMBL4227486)
Affinity DataIC50: 3nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461256(CHEMBL4228143)
Affinity DataIC50: 4nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461267(CHEMBL4227427)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461260(CHEMBL4228926)
Affinity DataIC50: 8nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461266(CHEMBL4226577)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461264(CHEMBL4227848)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461251(CHEMBL4228920)
Affinity DataIC50: 18nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461247(CHEMBL4228861)
Affinity DataIC50: 23nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461268(CHEMBL4225350)
Affinity DataIC50: 26nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461248(CHEMBL4227295)
Affinity DataIC50: 27nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461249(CHEMBL1215628)
Affinity DataIC50: 30nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461273(CHEMBL4227696)
Affinity DataIC50: 55nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461256(CHEMBL4228143)
Affinity DataIC50: 57nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461248(CHEMBL4227295)
Affinity DataIC50: 85nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461260(CHEMBL4228926)
Affinity DataIC50: 99nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum (isolate 3D7))
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461247(CHEMBL4228861)
Affinity DataIC50: 117nMAssay Description:Inhibition of Plasmodium falciparum falcipain-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461252(CHEMBL4224829)
Affinity DataIC50: 137nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461257(CHEMBL4228343)
Affinity DataIC50: 178nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461261(CHEMBL4229174)
Affinity DataIC50: 190nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461250(CHEMBL4227965)
Affinity DataIC50: 192nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461257(CHEMBL4228343)
Affinity DataIC50: 195nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461247(CHEMBL4228861)
Affinity DataIC50: 202nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461262(CHEMBL4226767)
Affinity DataIC50: 213nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461261(CHEMBL4229174)
Affinity DataIC50: 230nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461250(CHEMBL4227965)
Affinity DataIC50: 253nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461262(CHEMBL4226767)
Affinity DataIC50: 283nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461254(CHEMBL4225367)
Affinity DataIC50: 300nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461251(CHEMBL4228920)
Affinity DataIC50: 334nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461247(CHEMBL4228861)
Affinity DataIC50: 382nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461252(CHEMBL4224829)
Affinity DataIC50: 435nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461248(CHEMBL4227295)
Affinity DataIC50: 492nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461250(CHEMBL4227965)
Affinity DataIC50: 494nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461262(CHEMBL4226767)
Affinity DataIC50: 635nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFalcipain 2(malaria parasite P. falciparum)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461262(CHEMBL4226767)
Affinity DataIC50: 667nMAssay Description:Inhibition of Plasmodium falciparum falcipain-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin S(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461253(CHEMBL4228604)
Affinity DataIC50: 710nMAssay Description:Inhibition of human cathepsin SMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin B(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461255(CHEMBL4228800)
Affinity DataIC50: 715nMAssay Description:Inhibition of human cathepsin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461253(CHEMBL4228604)
Affinity DataIC50: 755nMAssay Description:Inhibition of human cathepsin LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCathepsin K(Human)
Irbm Science Park

Curated by ChEMBL
LigandPNGBDBM50461253(CHEMBL4228604)
Affinity DataIC50: 867nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
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