Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50002973
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.690nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465331(CHEMBL4294912)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465333(CHEMBL4287662)
Affinity DataIC50: 40nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465334(CHEMBL4288105)
Affinity DataIC50: 79nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465330(CHEMBL4277459)
Affinity DataIC50: 92nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465329(CHEMBL4279758)
Affinity DataIC50: 97nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465334(CHEMBL4288105)
Affinity DataIC50: 150nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465330(CHEMBL4277459)
Affinity DataIC50: 260nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465335(CHEMBL4280872)
Affinity DataIC50: 340nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465332(CHEMBL4284524)
Affinity DataIC50: 340nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465333(CHEMBL4287662)
Affinity DataIC50: 460nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465332(CHEMBL4284524)
Affinity DataIC50: 740nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465330(CHEMBL4277459)
Affinity DataIC50: 770nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465336(CHEMBL4284275)
Affinity DataIC50: 910nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465337(CHEMBL4291517)
Affinity DataIC50: 970nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465332(CHEMBL4284524)
Affinity DataIC50: 980nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465334(CHEMBL4288105)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465335(CHEMBL4280872)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465329(CHEMBL4279758)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of ROCK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465336(CHEMBL4284275)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465337(CHEMBL4291517)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465331(CHEMBL4294912)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465331(CHEMBL4294912)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of PKCalpha (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465337(CHEMBL4291517)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465333(CHEMBL4287662)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465335(CHEMBL4280872)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465329(CHEMBL4279758)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50465336(CHEMBL4284275)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed