Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002392
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50458056(CHEMBL4208031)
Affinity DataIC50: 107nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50458056(CHEMBL4208031)
Affinity DataIC50: 107nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50458055(CHEMBL4214605)
Affinity DataIC50: 136nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50458055(CHEMBL4214605)
Affinity DataIC50: 136nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50446143(CHEMBL3108897)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human LSD1/CoREST preincubated for 5 mins followed by ART-(N,N-dimethyl-K)-QTARKSTGGKAPRKQLA substrate addition measured af...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-2-phenylcyclopropanamine | cid_2723716 | (...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of MAO-B (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-2-phenylcyclopropanamine | cid_2723716 | (...)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of MAO-A (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50458055(CHEMBL4214605)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAO-B (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50458055(CHEMBL4214605)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of MAO-A (unknown origin) by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Medical University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50458057(CHEMBL4210908)
Affinity DataKi:  40nMAssay Description:Inhibition of LSD1/CoREST (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed