Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50001599
LigandPNGBDBM50263791(CHEMBL4062397)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human PDE2A1 using 3',5'-[3H]cGMP as substrate measured after 30 mins by Yttrium silicate scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
LigandPNGBDBM50286695(CHEMBL4160171)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human PDE2A1 using 3',5'-[3H]cGMP as substrate measured after 30 mins by Yttrium silicate scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
LigandPNGBDBM50286731(CHEMBL4171712)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human PDE2A1 using 3',5'-[3H]cGMP as substrate measured after 30 mins by Yttrium silicate scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
LigandPNGBDBM50263740(CHEMBL4088142)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of human PDE2A1 using 3',5'-[3H]cGMP as substrate measured after 30 mins by Yttrium silicate scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed
LigandPNGBDBM50263791(CHEMBL4062397)
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of PDE5A1 (unknown origin) using 3',5'-[3H]cGMP as substrate measured after 30 mins by Yttrium silicate scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2020
Entry Details Article
PubMed