Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50018906
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Shenzhen Salubris Pharmaceuticals Co.

Curated by ChEMBL
LigandPNGBDBM50613747(CHEMBL5280124)
Affinity DataIC50: 4.79E+3nMAssay Description:Antagonist activity at NOD1 in human HEK-Blue hNOD1 cells assessed as inhibition of C12-iE-DAP-induced SEAP release preincubated for 3 hrs followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetCytochrome P450 2C8(Human)
Shenzhen Salubris Pharmaceuticals Co.

Curated by ChEMBL
LigandPNGBDBM50613746(CHEMBL5271581)
Affinity DataIC50: 9.97E+3nMAssay Description:Inhibition of CYP2C8 in human liver microsomes using probe substrate in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Shenzhen Salubris Pharmaceuticals Co.

Curated by ChEMBL
LigandPNGBDBM50613747(CHEMBL5280124)
Affinity DataIC50: 1.31E+4nMAssay Description:Antagonist activity at NOD2 in human HEK-Blue hNOD2 cells assessed as inhibition of MDP-induced NOD2 activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed