Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50001500
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 0.452nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM23448(butyl 4-hydroxybenzoate | Nipabutyl | BUTYLPARABEN...)
Affinity DataIC50: 1.42E+3nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280387(CHEMBL4166909)
Affinity DataIC50: 7.98E+3nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280393(CHEMBL4170305)
Affinity DataIC50: 8.21E+3nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50240376(n-octylgallate | 3,4,5-Trihydroxy-benzoic acid oct...)
Affinity DataIC50: 8.74E+3nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280382(Butyl Gallate)
Affinity DataIC50: 8.97E+3nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280391(CHEMBL4169994)
Affinity DataIC50: 1.32E+4nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280390(CHEMBL4165518)
Affinity DataIC50: 1.62E+4nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280384(CHEMBL4163053)
Affinity DataIC50: 2.94E+4nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280392(CHEMBL4171348)
Affinity DataIC50: 3.25E+4nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280386(CHEMBL4174801)
Affinity DataIC50: 3.46E+4nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280385(CHEMBL4159672)
Affinity DataIC50: 3.94E+4nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280381(CHEMBL4173755)
Affinity DataIC50: 5.53E+4nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280389(CHEMBL4168938)
Affinity DataIC50: 6.04E+4nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280383(CHEMBL4163451)
Affinity DataIC50: 2.00E+5nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280388(CHEMBL4162076)
Affinity DataIC50: 2.00E+5nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Longwood University

Curated by ChEMBL
LigandPNGBDBM50280380(CHEMBL4160086)
Affinity DataIC50: 2.00E+5nMAssay Description:Displacement of Fluor.ES2 Green from human ERalpha by TR-FRET competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2020
Entry Details Article
PubMed