Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50001591
LigandPNGBDBM50286461(CHEMBL4166626)
Affinity DataIC50: 25nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286424(CHEMBL4170186)
Affinity DataIC50: 32nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286424(CHEMBL4170186)
Affinity DataIC50: 45nMAssay Description:Inhibition of p300/CBP in human PC3 cells assessed as reduction in acetylated H3K27 levels after 3 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286461(CHEMBL4166626)
Affinity DataIC50: 47nMAssay Description:Inhibition of p300/CBP in human PC3 cells assessed as reduction in acetylated H3K27 levels after 3 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286423(CHEMBL4174931)
Affinity DataIC50: 60nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286423(CHEMBL4174931)
Affinity DataIC50: 101nMAssay Description:Inhibition of p300/CBP in human PC3 cells assessed as reduction in acetylated H3K27 levels after 3 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286465(CHEMBL4177251)
Affinity DataIC50: 121nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286459(CHEMBL4163183)
Affinity DataIC50: 170nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286469(CHEMBL4173894)
Affinity DataIC50: 240nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286459(CHEMBL4163183)
Affinity DataIC50: 470nMAssay Description:Inhibition of p300/CBP in human PC3 cells assessed as reduction in acetylated H3K27 levels after 3 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286476(CHEMBL4168543)
Affinity DataIC50: 510nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286465(CHEMBL4177251)
Affinity DataIC50: 760nMAssay Description:Inhibition of p300/CBP in human PC3 cells assessed as reduction in acetylated H3K27 levels after 3 hrs by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286477(CHEMBL4167383)
Affinity DataIC50: 780nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50286423(CHEMBL4174931)
Affinity DataIC50: 990nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286466(CHEMBL4171897)
Affinity DataIC50: 990nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286464(CHEMBL4176737)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50286423(CHEMBL4174931)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286475(CHEMBL4167931)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286478(CHEMBL4160129)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286462(CHEMBL4175251)
Affinity DataIC50: 1.71E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286473(CHEMBL4171809)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286460(CHEMBL4176407)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286472(CHEMBL4168449)
Affinity DataIC50: 4.86E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286467(CHEMBL4161300)
Affinity DataIC50: 5.06E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286457(CHEMBL4159813)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286468(CHEMBL4165120)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286479(CHEMBL4164715)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286458(CHEMBL4170778)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286470(CHEMBL4168882)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286471(CHEMBL4160552)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Abbvie

Curated by ChEMBL
LigandPNGBDBM50286423(CHEMBL4174931)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed
LigandPNGBDBM50286463(CHEMBL4163946)
Affinity DataIC50: 2.78E+4nMAssay Description:Inhibition of p300/CBP (unknown origin) using biotinylated synthetic Histone H4 Peptide as substrate pretreated for 30 mins followed by substrate add...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2020
Entry Details Article
PubMed