Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50001660
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291820(CHEMBL4159155)
Affinity DataIC50: 0.290nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291735(CHEMBL4169891)
Affinity DataIC50: 0.330nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291816(CHEMBL4165983)
Affinity DataIC50: 0.380nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291733(CHEMBL4173065)
Affinity DataIC50: 0.460nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291734(CHEMBL4159247)
Affinity DataIC50: 0.580nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50162007(3-[(2R)-amino-2-phenylethyl]-1-(2,6-difluorobenzyl...)
Affinity DataIC50: 0.590nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291819(CHEMBL4170478)
Affinity DataIC50: 0.740nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291825(CHEMBL4167067)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291741(CHEMBL4161566)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291734(CHEMBL4159247)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291833(CHEMBL4163619)
Affinity DataIC50: 2.30nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291740(CHEMBL4169486)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rhesus macaque)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291734(CHEMBL4159247)
Affinity DataIC50: 3.5nMAssay Description:Displacement of [125I]D-Trp6-LHRH from monkey GnRH receptor expressed in HEK293 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rhesus macaque)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291733(CHEMBL4173065)
Affinity DataIC50: 3.80nMAssay Description:Displacement of [125I]D-Trp6-LHRH from monkey GnRH receptor expressed in HEK293 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rhesus macaque)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291735(CHEMBL4169891)
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]D-Trp6-LHRH from monkey GnRH receptor expressed in HEK293 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291735(CHEMBL4169891)
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291817(CHEMBL4173914)
Affinity DataIC50: 5.40nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291764(CHEMBL4160683)
Affinity DataIC50: 6.20nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291733(CHEMBL4173065)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291813(CHEMBL4169027)
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291739(CHEMBL4176683)
Affinity DataIC50: 8.40nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291742(CHEMBL4172886)
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291808(CHEMBL4171288)
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291809(CHEMBL4175801)
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291738(CHEMBL4166067)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291812(CHEMBL4164508)
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291752(CHEMBL4166009)
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291814(CHEMBL4161096)
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291818(CHEMBL4162543)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291743(CHEMBL4169864)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291744(CHEMBL4164522)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291736(CHEMBL4162619)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291750(CHEMBL4174753)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291811(CHEMBL4172391)
Affinity DataIC50: 46nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291829(CHEMBL4164417)
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291810(CHEMBL4167945)
Affinity DataIC50: 62nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291737(CHEMBL4173316)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291827(CHEMBL4170863)
Affinity DataIC50: 69nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291826(CHEMBL4174298)
Affinity DataIC50: 73nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291749(CHEMBL4160698)
Affinity DataIC50: 89nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291830(CHEMBL4175063)
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291748(CHEMBL4171296)
Affinity DataIC50: 142nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291745(CHEMBL4172405)
Affinity DataIC50: 144nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291747(CHEMBL4175816)
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291832(CHEMBL4173938)
Affinity DataIC50: 165nMAssay Description:Antagonist activity at human GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50291735(CHEMBL4169891)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at rat GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced NF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50291733(CHEMBL4173065)
Affinity DataIC50: 279nMAssay Description:Antagonist activity at rat GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced NF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50291734(CHEMBL4159247)
Affinity DataIC50: 590nMAssay Description:Antagonist activity at rat GnRH receptor expressed in HEK293 cells co-expressing pGL4-NFATpromoter AP-1-luc assessed as inhibition of GnRH-induced NF...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291828(CHEMBL4160259)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Tiumbio

Curated by ChEMBL
LigandPNGBDBM50291831(CHEMBL4172747)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]D-Trp6-LHRH from human GnRH receptor expressed in CHO-K1 cells after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2020
Entry Details Article
PubMed
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