Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50001583
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286229(CHEMBL4167612)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286068(CHEMBL4171201)
Affinity DataEC50:  5.80E+3nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataEC50:  7.90E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286246(CHEMBL4159695)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286247(CHEMBL4164159)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286230(CHEMBL4171371)
Affinity DataEC50:  1.40E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286248(CHEMBL4168030)
Affinity DataEC50:  4.20E+3nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286251(CHEMBL4167844)
Affinity DataEC50:  9.30E+3nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286249(CHEMBL4159929)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286231(CHEMBL4175056)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286245(CHEMBL4163070 | US11981669, Comparative Example 1)
Affinity DataEC50:  1.90E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286070(CHEMBL4166512)
Affinity DataEC50:  1.50E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286233(CHEMBL4175892)
Affinity DataEC50:  5.80E+3nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286232(CHEMBL4173606)
Affinity DataEC50:  1.40E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286250(CHEMBL4159751)
Affinity DataEC50:  5.80E+3nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286228(CHEMBL4174643)
Affinity DataEC50:  4.50E+3nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286224(CHEMBL4162891)
Affinity DataEC50:  1.70E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286072(CHEMBL4164403)
Affinity DataEC50:  4.70E+3nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286227(CHEMBL4160770)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286069(CHEMBL4174815)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286263(CHEMBL4167657)
Affinity DataEC50:  1.30E+4nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286071(CHEMBL4166742)
Affinity DataEC50:  5.70E+3nMAssay Description:Inhibition of PHD2 in human Hep3B cells assessed as increase in EPO release after 24 hrs by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286250(CHEMBL4159751)
Affinity DataIC50: 110nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286228(CHEMBL4174643)
Affinity DataIC50: 120nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286232(CHEMBL4173606)
Affinity DataIC50: 190nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286231(CHEMBL4175056)
Affinity DataIC50: 210nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286071(CHEMBL4166742)
Affinity DataIC50: 220nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286068(CHEMBL4171201)
Affinity DataIC50: 290nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 300nMAssay Description:Inhibition of PHD2 (181 to 426 residues) (unknown origin) using biotinylated CODD peptide as substrate preincubated for 15 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286263(CHEMBL4167657)
Affinity DataIC50: 370nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286233(CHEMBL4175892)
Affinity DataIC50: 450nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286227(CHEMBL4160770)
Affinity DataIC50: 650nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286224(CHEMBL4162891)
Affinity DataIC50: 720nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286072(CHEMBL4164403)
Affinity DataIC50: 730nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286230(CHEMBL4171371)
Affinity DataIC50: 730nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286069(CHEMBL4174815)
Affinity DataIC50: 820nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286248(CHEMBL4168030)
Affinity DataIC50: 850nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286247(CHEMBL4164159)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286070(CHEMBL4166512)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286245(CHEMBL4163070 | US11981669, Comparative Example 1)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286251(CHEMBL4167844)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286246(CHEMBL4159695)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286249(CHEMBL4159929)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50193145(Isoquinoline 3 | CHEMBL426560 | N-[(1-CHLORO-4-HYD...)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEgl nine homolog 1(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286229(CHEMBL4167612)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human HIF-PHD2 assessed as reduction in HIF1-alpha binding to VBC complex using biotin-labeled HIF1-alpha peptide as substrate preincub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCytochrome P450 2A6(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286071(CHEMBL4166742)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP2A6 in human liver microsomes by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCytochrome P450 2C8(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286071(CHEMBL4166742)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP2C8 in human liver microsomes by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
LigandPNGBDBM50286071(CHEMBL4166742)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ERG expressed in HEK293 cells at holding potential of -80 mV by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCytochrome P450 2B6(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286071(CHEMBL4166742)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP2B6 in human liver microsomes by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Japan Tobacco

Curated by ChEMBL
LigandPNGBDBM50286071(CHEMBL4166742)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CYP1A2 in human liver microsomes by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2020
Entry Details Article
PubMed
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