Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50002140
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454051(CHEMBL4207636)
Affinity DataIC50: 1.66E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454049(CHEMBL4214332)
Affinity DataIC50: 1.84E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454048(CHEMBL4213826)
Affinity DataIC50: 2.66E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50099585(1-[4-(2-Azepan-1-yl-ethoxy)-benzyl]-2-(4-hydroxy-p...)
Affinity DataIC50: 3.17E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454053(CHEMBL4203135)
Affinity DataIC50: 5.12E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454050(CHEMBL4209434)
Affinity DataIC50: 5.50E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454057(CHEMBL4218272)
Affinity DataIC50: 6.08E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454055(CHEMBL4207948)
Affinity DataIC50: 6.11E+4nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454056(CHEMBL4215448)
Affinity DataIC50: 3.56E+5nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454052(CHEMBL4206393)
Affinity DataIC50: 4.82E+5nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Central University of Punjab

Curated by ChEMBL
LigandPNGBDBM50454054(CHEMBL4218756)
Affinity DataIC50: 5.87E+5nMAssay Description:Displacement of Fluormone-tagged ES2 from human recombinant ERalpha after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed