Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50035791
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM91718(Androst-1,4-dien-3,17-dione, 7)
Affinity DataKi:  120nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataKi:  220nMAssay Description:Competitive inhibition of binding to human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM91718(Androst-1,4-dien-3,17-dione, 7)
Affinity DataKi:  260nMAssay Description:Inactivation rate (Ki) for human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50014314(9a,11a-Dimethyl-3a,4,5,9a,9b,10,11,11a-octahydro-3...)
Affinity DataKi:  390nMAssay Description:Inactivation rate (Ki) for human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50014314(9a,11a-Dimethyl-3a,4,5,9a,9b,10,11,11a-octahydro-3...)
Affinity DataKi:  410nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020640(CHEMBL349300 | 10,13-Dimethyl-6,7,8,9,10,11,12,13,...)
Affinity DataKi:  690nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020640(CHEMBL349300 | 10,13-Dimethyl-6,7,8,9,10,11,12,13,...)
Affinity DataKi:  1.10E+3nMAssay Description:Inactivation rate (Ki) of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataKi:  1.55E+3nMAssay Description:Inactivation rate (Ki) of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020645(CHEMBL158600 | 2,4b-Dimethyl-7-oxo-1,2,3,4,4a,4b,7...)
Affinity DataKi:  3.98E+3nMAssay Description:Inactivation rate (Ki) of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020647(CHEMBL348154 | 7-Hydroxymethyl-4a,7-dimethyl-4b,5,...)
Affinity DataKi:  8.56E+3nMAssay Description:Inactivation rate (Ki) of human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020641(CHEMBL158397 | Acetic acid 2,4b-dimethyl-7-oxo-1,2...)
Affinity DataKi:  1.30E+4nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020639(CHEMBL158326 | 7-Acetyl-4a,7-dimethyl-4b,5,6,7,8,8...)
Affinity DataKi:  4.50E+4nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020642(CHEMBL158325 | 4a,7-Dimethyl-7-propionyl-4b,5,6,7,...)
Affinity DataKi:  9.70E+4nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020644(CHEMBL423772 | 1,2,4b-Trimethyl-7-oxo-1,2,3,4,4a,4...)
Affinity DataKi:  1.03E+5nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020643(CHEMBL346929 | 2,4b-Dimethyl-7-oxo-1,2,3,4,4a,4b,7...)
Affinity DataKi:  1.30E+5nMAssay Description:Competitive inhibition of binding to human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020638(CHEMBL158717 | 2,4b-Dimethyl-7-oxo-1,2,3,4,4a,4b,7...)
Affinity DataKi:  8.93E+5nMAssay Description:Competitive inhibition of binding to human placental aromatase Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed
TargetAromatase(Human)
Washington University

Curated by ChEMBL
LigandPNGBDBM50020646(CHEMBL160271 | 1,2,4b-Trimethyl-7-oxo-1,2,3,4,4a,4...)
Affinity DataKi:  1.20E+6nMAssay Description:Competitive inhibition of binding to human placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2012
Entry Details Article
PubMed