Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002134
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 10nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453941(CHEMBL4210489)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453940(CHEMBL4209034)
Affinity DataIC50: 3.05E+3nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453943(CHEMBL509962)
Affinity DataIC50: 3.34E+3nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453936(CHEMBL4216885)
Affinity DataIC50: 3.88E+3nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453937(CHEMBL4212655)
Affinity DataIC50: 6.87E+3nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453942(CHEMBL469266 | INF-55)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453939(CHEMBL4207850)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM67905(SMR000179854 | MLS000546456 | 5-chloranyl-2-phenyl...)
Affinity DataIC50: 2.28E+4nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAromatase(Human)
University of Hawai'I At Hilo

Curated by ChEMBL
LigandPNGBDBM50453938(CHEMBL4204862)
Affinity DataIC50: 3.97E+4nMAssay Description:Inhibition of CYP19A1 (unknown origin) preincubated with NADPH followed by DBF substrate addition after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed