Compile Data Set for Download or QSAR
Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50001548
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM39862(Selegiline | MLS000069378 | N-methyl-1-phenyl-N-pr...)
Affinity DataIC50: 20nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283860(CHEMBL4169543)
Affinity DataIC50: 110nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283916(CHEMBL1782842)
Affinity DataIC50: 120nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283866(CHEMBL475017)
Affinity DataIC50: 177nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283933(CHEMBL4163328)
Affinity DataIC50: 210nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283915(CHEMBL4167042)
Affinity DataIC50: 240nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283855(CHEMBL4167829)
Affinity DataIC50: 270nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283915(CHEMBL4167042)
Affinity DataIC50: 290nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283851(CHEMBL4167325)
Affinity DataIC50: 290nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283866(CHEMBL475017)
Affinity DataIC50: 310nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283853(CHEMBL4172849)
Affinity DataIC50: 320nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283802(CHEMBL4176805)
Affinity DataIC50: 330nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283801(CHEMBL475188)
Affinity DataIC50: 350nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283934(CHEMBL4165825)
Affinity DataIC50: 380nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283800(CHEMBL4164943)
Affinity DataIC50: 440nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283865(CHEMBL4169131)
Affinity DataIC50: 640nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283853(CHEMBL4172849)
Affinity DataIC50: 760nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283852(CHEMBL1782829)
Affinity DataIC50: 760nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283950(CHEMBL4173275)
Affinity DataIC50: 920nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283907(CHEMBL4161683)
Affinity DataIC50: 960nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283848(CHEMBL4163586)
Affinity DataIC50: 990nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283855(CHEMBL4167829)
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283806(CHEMBL4166188)
Affinity DataIC50: 1.22E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283916(CHEMBL1782842)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283949(CHEMBL1782841)
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283804(CHEMBL4166029)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283857(CHEMBL471758)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283885(CHEMBL470744)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283913(CHEMBL4176387)
Affinity DataIC50: 2.08E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283806(CHEMBL4166188)
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283933(CHEMBL4163328)
Affinity DataIC50: 2.97E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283860(CHEMBL4169543)
Affinity DataIC50: 3.33E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283935(CHEMBL4167525)
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283849(CHEMBL4169612)
Affinity DataIC50: 4.24E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283949(CHEMBL1782841)
Affinity DataIC50: 4.33E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283947(CHEMBL4161532)
Affinity DataIC50: 4.85E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283864(CHEMBL471769)
Affinity DataIC50: 5.07E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283856(CHEMBL4165104)
Affinity DataIC50: 5.07E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283885(CHEMBL470744)
Affinity DataIC50: 5.76E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283908(CHEMBL4173005)
Affinity DataIC50: 5.78E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283890(CHEMBL4171487)
Affinity DataIC50: 6.04E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283862(CHEMBL4169453)
Affinity DataIC50: 6.12E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283861(CHEMBL4177110)
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283861(CHEMBL4177110)
Affinity DataIC50: 7.14E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283865(CHEMBL4169131)
Affinity DataIC50: 7.48E+3nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283934(CHEMBL4165825)
Affinity DataIC50: 8.61E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283857(CHEMBL471758)
Affinity DataIC50: 8.86E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283808(CHEMBL4171408)
Affinity DataIC50: 9.31E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Government College University

Curated by ChEMBL
LigandPNGBDBM50283864(CHEMBL471769)
Affinity DataIC50: 9.47E+3nMAssay Description:Inhibition of MAO-B in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMed
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