Compile Data Set for Download or QSAR
Report error Found 92 Enz. Inhib. hit(s) with all data for entry = 50000256
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243627(CHEMBL4068708)
Affinity DataIC50: 0.610nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243612(CHEMBL4093165)
Affinity DataIC50: 0.631nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243627(CHEMBL4068708)
Affinity DataIC50: 0.631nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243612(CHEMBL4093165)
Affinity DataIC50: 0.660nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243645(CHEMBL4087520)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243645(CHEMBL4087520)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243561(CHEMBL4086535)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243625(CHEMBL4094098)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243589(CHEMBL4095223)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243608(CHEMBL4100882)
Affinity DataIC50: 1.26nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243561(CHEMBL4086535)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243588(CHEMBL4067800)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243589(CHEMBL4095223)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243593(CHEMBL4089947)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243608(CHEMBL4100882)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243588(CHEMBL4067800)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243593(CHEMBL4089947)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243625(CHEMBL4094098)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243536(CHEMBL4062749)
Affinity DataIC50: 1.58nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243626(CHEMBL4089821)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243609(CHEMBL4090706)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243536(CHEMBL4062749)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243626(CHEMBL4089821)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243609(CHEMBL4090706)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243637(CHEMBL4068853)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243535(CHEMBL4065097)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243644(CHEMBL4066563)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243637(CHEMBL4068853)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243535(CHEMBL4065097)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243644(CHEMBL4066563)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243594(CHEMBL4082908)
Affinity DataIC50: 2.5nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243594(CHEMBL4082908)
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243587(CHEMBL4105382)
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243587(CHEMBL4105382)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243610(CHEMBL4063825)
Affinity DataIC50: 3.80nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243610(CHEMBL4063825)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243547(CHEMBL4076020)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243547(CHEMBL4076020)
Affinity DataIC50: 5.01nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243545(CHEMBL4078689)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243545(CHEMBL4078689)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243611(CHEMBL4085407)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243611(CHEMBL4085407)
Affinity DataIC50: 6.31nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243560(CHEMBL4102969)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243560(CHEMBL4102969)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243546(CHEMBL4072418)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243546(CHEMBL4072418)
Affinity DataIC50: 83nMAssay Description:Antagonist activity at recombinant human CB1 receptor expressed in HEK293 cell membranes assessed as inhibition of CP55940-induced [35S]GTPgammaS bin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243536(CHEMBL4062749)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in beta-galactosidase expressing CHOK1 cell membranes after 60 mins by scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243536(CHEMBL4062749)
Affinity DataKi:  0.0100nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in beta-galactosidase expressing CHOK1 cell membranes after 60 mins by scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243589(CHEMBL4095223)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in beta-galactosidase expressing CHOK1 cell membranes after 60 mins by scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50243589(CHEMBL4095223)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in beta-galactosidase expressing CHOK1 cell membranes after 60 mins by scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2019
Entry Details Article
PubMed
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