Compile Data Set for Download or QSAR
Report error Found 135 Enz. Inhib. hit(s) with all data for entry = 50002886
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464401(CHEMBL4288690)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464403(CHEMBL4294790)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464410(CHEMBL4292109)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464404(CHEMBL4286494)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464411(CHEMBL4291381)
Affinity DataEC50:  0.700nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464400(CHEMBL4293386)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464412(CHEMBL4278248)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464407(CHEMBL4292336)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464406(CHEMBL4280601)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464404(CHEMBL4286494)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464420(CHEMBL4290302)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464421(CHEMBL4286896)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464403(CHEMBL4294790)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464399(CHEMBL4278446)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464416(CHEMBL4289115)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464417(CHEMBL4280791)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464422(CHEMBL4277390)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464418(CHEMBL4284223)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464412(CHEMBL4278248)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464407(CHEMBL4292336)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464408(CHEMBL4285145)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464421(CHEMBL4286896)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464416(CHEMBL4289115)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464417(CHEMBL4280791)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464410(CHEMBL4292109)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464401(CHEMBL4288690)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464400(CHEMBL4293386)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464406(CHEMBL4280601)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464409(CHEMBL4283539)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464418(CHEMBL4284223)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464413(CHEMBL4281712)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464402(CHEMBL4279639)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464411(CHEMBL4291381)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464405(CHEMBL4281915)
Affinity DataEC50:  8nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464415(CHEMBL4278575)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464420(CHEMBL4290302)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464422(CHEMBL4277390)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464415(CHEMBL4278575)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464406(CHEMBL4280601)
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1A(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464412(CHEMBL4278248)
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464412(CHEMBL4278248)
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464415(CHEMBL4278575)
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 135 total ) | Next | Last >>
Jump to: