Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50002003
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451951(CHEMBL4217941)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451934(CHEMBL4207594)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451935(CHEMBL4208825)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451931(CHEMBL4213552)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451962(CHEMBL4214058)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451932(CHEMBL4204793)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 13nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451948(CHEMBL4209658)
Affinity DataIC50: 14nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451938(CHEMBL4207152)
Affinity DataIC50: 16nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451937(CHEMBL4210581)
Affinity DataIC50: 17nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451949(CHEMBL4218884)
Affinity DataIC50: 17nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM85573(7-Hydroxy-flavone, 5h)
Affinity DataIC50: 35nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50049402(2-(3,4-dimethoxyphenyl)-7-hydroxy-4H-chromen-4-one...)
Affinity DataIC50: 37nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50025480(NSC-127572 | CHEMBL485247)
Affinity DataIC50: 44nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451961(CHEMBL4205720)
Affinity DataIC50: 48nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451936(CHEMBL4216881)
Affinity DataIC50: 57nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451950(CHEMBL4203490)
Affinity DataIC50: 66nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50451933(CHEMBL4218485)
Affinity DataIC50: 67nMAssay Description:Inhibition of rat brain AChE using acetylthiocholine iodide as substrate by spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed