Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50001540
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283680(CHEMBL4164470)
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283674(CHEMBL4176578)
Affinity DataIC50: 0.540nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283666(CHEMBL4169845)
Affinity DataIC50: 0.610nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283675(CHEMBL4175111)
Affinity DataIC50: 0.720nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283673(CHEMBL4165967)
Affinity DataIC50: 0.760nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283543(CHEMBL4172793)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283678(CHEMBL4162971)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283671(CHEMBL4169403)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283672(CHEMBL4164893)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50335784(2-[6-(3-Aminopiperidin-1-yl)-3-methyl-2,4-dioxo-3,...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283677(CHEMBL4173673)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283544(CHEMBL4173272)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283630(CHEMBL4161924)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283664(CHEMBL4161474)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283676(CHEMBL4165359)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283545(CHEMBL4162340)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283668(CHEMBL4169618)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283669(CHEMBL4177478)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283670(CHEMBL4174924)
Affinity DataIC50: 15nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283576(CHEMBL4162532)
Affinity DataIC50: 18nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283665(CHEMBL4173215)
Affinity DataIC50: 27nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283667(CHEMBL4165788)
Affinity DataIC50: 100nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283679(CHEMBL4173013)
Affinity DataIC50: 100nMAssay Description:Inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283545(CHEMBL4162340)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of DPP9 (unknown origin) using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283545(CHEMBL4162340)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of DPP8 (unknown origin) using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50283545(CHEMBL4162340)
Affinity DataKi:  2.90nMAssay Description:Reversible mixed-type inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
The First Affiliated Hospital of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50335784(2-[6-(3-Aminopiperidin-1-yl)-3-methyl-2,4-dioxo-3,...)
Affinity DataKi:  5.10nMAssay Description:Competitive inhibition of human DPP4 using Gly-Pro-AMC as substrate preincubated for 10 mins followed by substrate addition measured for 5 to 10 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)