Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50001421
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279227(CHEMBL4167203)
Affinity DataKd: <1.00E+3nMAssay Description:Binding affinity to recombinant N-terminal domain of human 15N-labeled MDM2 (1 to 118 residues) at Arg29 residue expressed in Escherichia coli BL21-C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279230(CHEMBL4170591)
Affinity DataKi:  80nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279223(CHEMBL4177057)
Affinity DataKi:  90nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279228(CHEMBL4171622)
Affinity DataKi:  100nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279227(CHEMBL4167203)
Affinity DataKi:  140nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279253(CHEMBL4176936)
Affinity DataKi:  320nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279232(CHEMBL4177390)
Affinity DataKi:  340nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279224(CHEMBL4169074)
Affinity DataKi:  350nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279254(CHEMBL4160424)
Affinity DataKi:  600nMAssay Description:Displacement of fluorescent-labelled P4 peptide from recombinant human MDM2 expressed in Escherichia coli BL21(DE3) Rosetta after 30 mins by fluoresc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279234(CHEMBL4169196)
Affinity DataKi:  700nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279235(CHEMBL4159944)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279225(CHEMBL4175068)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279231(CHEMBL4166759)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279226(CHEMBL4167652)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279233(CHEMBL4175521)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Human)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50279229(CHEMBL4168287)
Affinity DataKi:  5.30E+3nMAssay Description:Displacement of 5'FAM-LTFEHYWAQLTS from recombinant human N-terminal MDM2 (1 to 118 residues) expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed