Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50000884
TargetKelch-like ECH-associated protein 1(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50262959(CHEMBL4083845)
Affinity DataIC50: 160nMAssay Description:Binding affinity to His-tagged Keap1 DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli assessed as reduction in protein ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50262960(CHEMBL4099355)
Affinity DataIC50: 170nMAssay Description:Binding affinity to His-tagged Keap1 DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli assessed as reduction in protein ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50262957(CHEMBL4091619)
Affinity DataIC50: 180nMAssay Description:Binding affinity to His-tagged Keap1 DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli assessed as reduction in protein ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50262955(CHEMBL4077198)
Affinity DataIC50: 200nMAssay Description:Binding affinity to His-tagged Keap1 DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli assessed as reduction in protein ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50006932(CHEMBL3237245)
Affinity DataIC50: 230nMAssay Description:Binding affinity to His-tagged Keap1 DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli assessed as reduction in protein ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50262958(CHEMBL4070735)
Affinity DataIC50: 260nMAssay Description:Binding affinity to His-tagged Keap1 DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli assessed as reduction in protein ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50262956(CHEMBL4062108)
Affinity DataIC50: 290nMAssay Description:Binding affinity to His-tagged Keap1 DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli assessed as reduction in protein ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Keio University

Curated by ChEMBL
LigandPNGBDBM50006931(CHEMBL2402207)
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity to His-tagged Keap1 DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli assessed as reduction in protein ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/27/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)