Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50018904
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613736(CHEMBL3359320)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613736(CHEMBL3359320)
Affinity DataIC50: 4.50E+3nMAssay Description:Allosteric inhibition of H+ ATPase pma1 isoform by measuring NADP-coupled ATPase activity in presence of 1 mM ATP by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613731(CHEMBL5270653)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613736(CHEMBL3359320)
Affinity DataIC50: 6.30E+3nMAssay Description:Allosteric inhibition of H+ ATPase pma1 isoform by measuring NADP-coupled ATPase activity in presence of 10 mM ATP by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613727(CHEMBL4548520)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613728(CHEMBL4289313)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613732(CHEMBL5273581)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613744(CHEMBL5267780)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613727(CHEMBL4548520)
Affinity DataIC50: 1.68E+4nMAssay Description:Allosteric inhibition of H+ ATPase pma1 isoform by measuring NADP-coupled ATPase activity in presence of 10 mM ATP by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613733(CHEMBL4871324)
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613743(CHEMBL5268677)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613730(CHEMBL4518197)
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613742(CHEMBL5286133)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613729(CHEMBL5282411)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613745(CHEMBL5282994)
Affinity DataIC50: 2.49E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613727(CHEMBL4548520)
Affinity DataIC50: 2.97E+4nMAssay Description:Allosteric inhibition of H+ ATPase pma1 isoform by measuring NADP-coupled ATPase activity in presence of 1 mM ATP by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613740(CHEMBL5282214)
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613741(CHEMBL5287997)
Affinity DataIC50: 5.18E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613734(CHEMBL5277475)
Affinity DataIC50: 5.27E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613729(CHEMBL5282411)
Affinity DataIC50: 6.00E+4nMAssay Description:Allosteric inhibition of H+ ATPase pma1 isoform by measuring NADP-coupled ATPase activity in presence of 10 mM ATP by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613729(CHEMBL5282411)
Affinity DataIC50: 7.80E+4nMAssay Description:Allosteric inhibition of H+ ATPase pma1 isoform by measuring NADP-coupled ATPase activity in presence of 1 mM ATP by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613735(CHEMBL5278473)
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613739(CHEMBL5282458)
Affinity DataIC50: 1.67E+5nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613738(CHEMBL5278886)
Affinity DataIC50: 1.67E+5nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetThyrotropin receptor(Rat)
Pcovery

Curated by ChEMBL
LigandPNGBDBM50613737(CHEMBL5290293)
Affinity DataIC50: 1.67E+5nMAssay Description:Inhibition of Saccharomyces cerevisiae H+ ATPase pma1 isoform assessed as ATP hydrolysis incubated for 30 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed