Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50002057
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50002338(10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsul...)
Affinity DataIC50: 2.80nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50002338(10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsul...)
Affinity DataIC50: 17nMAssay Description:Affinity for displacement of [3H]WB-4101 labeled Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50001884(8-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)
Affinity DataIC50: 38nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019909(N-[(3-Chloro-phenyl)-(5-hydroxy-1,3-dimethyl-1H-py...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019916(2,2-Dichloro-N-[(3-chloro-phenyl)-(5-hydroxy-1,3-d...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50002338(10-[2-(1-Methyl-piperidin-2-yl)-ethyl]-2-methylsul...)
Affinity DataIC50: 1.30E+3nMAssay Description:Affinity for displacement of [3H]clonidine labeled Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019912(4-[(4-Fluoro-phenyl)-imino-methyl]-2,5-dimethyl-2H...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019913(4-[(3-Chloro-phenyl)-imino-methyl]-2,5-dimethyl-2H...)
Affinity DataIC50: 1.00E+4nMAssay Description:Affinity for displacement of [3H]clonidine labeled Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019914(4-[(3-Bromo-phenyl)-imino-methyl]-2,5-dimethyl-2H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019915(4-[(3-Chloro-phenyl)-imino-methyl]-2-isopropyl-5-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019913(4-[(3-Chloro-phenyl)-imino-methyl]-2,5-dimethyl-2H...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019911(2-Ethyl-4-(imino-phenyl-methyl)-5-methyl-2H-pyrazo...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019918(4-[(3-Chloro-phenyl)-imino-methyl]-5-methyl-2-prop...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019917(4-[Imino-(4-trifluoromethyl-phenyl)-methyl]-2,5-di...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019910(4-(Imino-phenyl-methyl)-2,5-dimethyl-2H-pyrazol-3-...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019920(4-[(3-Fluoro-phenyl)-imino-methyl]-2,5-dimethyl-2H...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019919(N-[(3-Chloro-phenyl)-(5-hydroxy-1,3-dimethyl-1H-py...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019913(4-[(3-Chloro-phenyl)-imino-methyl]-2,5-dimethyl-2H...)
Affinity DataIC50: 1.00E+4nMAssay Description:Affinity for displacement of [3H]SCH-23390 labeled Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019913(4-[(3-Chloro-phenyl)-imino-methyl]-2,5-dimethyl-2H...)
Affinity DataIC50: 1.00E+4nMAssay Description:Affinity for displacement of [3H]WB-4101 labeled Dopamine receptor D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Warner-Lambert/Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50019908(4-[(3-Chloro-phenyl)-imino-methyl]-2-ethyl-5-methy...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro binding affinity against Dopamine receptor D2 by displacement of [3H]haloperidol from rat striatal membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed