Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50048736
LigandPNGBDBM50226239(CHEMBL50451)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226234(CHEMBL50979)
Affinity DataKi:  0.160nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226227(CHEMBL52155)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226235(CHEMBL54288)
Affinity DataKi:  0.180nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226233(CHEMBL275524)
Affinity DataKi:  0.190nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.190nMAssay Description:Binding affinity against alpha-1-adrenoceptor was determined by displacement of [3H]-prazosin in rat brain homogenates.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226237(CHEMBL299584)
Affinity DataKi:  0.240nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226229(CHEMBL52439)
Affinity DataKi:  0.260nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226225(CHEMBL50746)
Affinity DataKi:  0.270nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226228(CHEMBL50137)
Affinity DataKi:  0.270nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226238(CHEMBL301614)
Affinity DataKi:  0.290nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226241(CHEMBL301749)
Affinity DataKi:  0.310nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226230(CHEMBL50084)
Affinity DataKi:  0.320nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226242(CHEMBL51056)
Affinity DataKi:  0.360nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226231(CHEMBL50473)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226232(CHEMBL300972)
Affinity DataKi:  0.470nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226236(CHEMBL300632)
Affinity DataKi:  0.870nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226240(CHEMBL298946)
Affinity DataKi:  0.920nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM50226226(CHEMBL422581)
Affinity DataKi:  1.70nMAssay Description:Binding affinity against alpha-1-adrenoceptor in rat brain homogenates [3H]-prazosin displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  4.83E+3nMAssay Description:Binding affinity against alpha-2-adrenoceptor was determined by displacement of [3H]-clonidine in rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2018
Entry Details Article
PubMed