Compile Data Set for Download or QSAR
Report error Found 139 Enz. Inhib. hit(s) with all data for entry = 50019108
TargetInterleukin-1 receptor-associated kinase 4(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615358(CHEMBL5282803)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human GST-tagged IRAK4 incubated for 30 mins in presence of ATP by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50076185(CHEMBL3416026 | US9290481, 1.1)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211951(US9290481, 1.2)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211952(US9290481, 1.3)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50076187(CHEMBL3416027 | US9290481, 1.4)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211953(US9290481, 2.1)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211954(US9290481, 2.2)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211955(US9290481, 2.3)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211956(US9290481, 2.4)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211957(US9290481, 2.5)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211958(US9290481, 2.6)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SYK using 5-Fluo-Ahx-GAPDYENLQELNKK-Amid as substrate in presence of ATP by microfluidic mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615314(CHEMBL5270667)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615315(CHEMBL5275887)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615316(CHEMBL5272249)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615317(CHEMBL5271126)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615318(CHEMBL5269901)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615319(CHEMBL5282393)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615320(CHEMBL5281109)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615321(CHEMBL5288239)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615322(CHEMBL5287305)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615323(CHEMBL5270834)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615324(CHEMBL5274905)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615325(CHEMBL5285217)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615326(CHEMBL5278557)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615327(CHEMBL5282609)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615328(CHEMBL5289952)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615329(CHEMBL5268696)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615330(CHEMBL5273906)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615331(CHEMBL5280041)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615332(CHEMBL5276953)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615333(CHEMBL5266175)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615334(CHEMBL5270622)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615335(CHEMBL5272817)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615336(CHEMBL5272260)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615337(CHEMBL5282796)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPolycomb complex protein BMI-1(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615338(CHEMBL5278972)
Affinity DataIC50: 1nMAssay Description:Inhibition of BMI1 (unknown origin) by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615357(CHEMBL5266861)
Affinity DataIC50: 1nMAssay Description:Inhibition of human GST-tagged IRAK4 incubated for 30 mins in presence of ATP by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM311561(US10155765, Example 59 | 2-[(2- aminoethyl)amino]-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human GST-tagged IRAK4 incubated for 30 mins in presence of ATP by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615356(CHEMBL5283042)
Affinity DataIC50: 3nMAssay Description:Inhibition of human GST-tagged IRAK4 incubated for 30 mins in presence of ATP by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetInterleukin-1 receptor-associated kinase 4(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM311562(US10155765, Example 60 | 2-[(2- aminoethyl)amino]-...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human GST-tagged IRAK4 incubated for 30 mins in presence of ATP by fluorescent polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615309(CHEMBL5285888)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615310(CHEMBL5278558)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615311(CHEMBL5288780)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50615312(CHEMBL5287185)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM5718(2,6,9-Trisubstituted purine deriv. 26 | 2-{[6-(ben...)
Affinity DataIC50: 5nMAssay Description:Inhibition of CDK2/cyclin E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50076185(CHEMBL3416026 | US9290481, 1.1)
Affinity DataIC50: 14nMAssay Description:Inhibition of SYK in human Ramos cells assessed as reduction in anti IgM-induced phosphorylation of BLNK by flow cytometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211951(US9290481, 1.2)
Affinity DataIC50: 14nMAssay Description:Inhibition of SYK in human Ramos cells assessed as reduction in anti IgM-induced phosphorylation of BLNK by flow cytometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211952(US9290481, 1.3)
Affinity DataIC50: 14nMAssay Description:Inhibition of SYK in human Ramos cells assessed as reduction in anti IgM-induced phosphorylation of BLNK by flow cytometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM50076187(CHEMBL3416027 | US9290481, 1.4)
Affinity DataIC50: 14nMAssay Description:Inhibition of SYK in human Ramos cells assessed as reduction in anti IgM-induced phosphorylation of BLNK by flow cytometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Universita Degli Studi Di Palermo

Curated by ChEMBL
LigandPNGBDBM211953(US9290481, 2.1)
Affinity DataIC50: 14nMAssay Description:Inhibition of SYK in human Ramos cells assessed as reduction in anti IgM-induced phosphorylation of BLNK by flow cytometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
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