Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50048743
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to membrane preparation from rat lung reticulocyte pretreated with alkylating beta-blocker...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKd:  1nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKd:  2nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding sites on beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating beta-blo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKd:  1.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating beta-blo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKd:  1.20nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKd:  2.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKi:  0.460nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKi:  0.610nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKi:  1.80nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKi:  2.80nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKi:  4.5nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKi:  20nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKi:  23nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKi:  31nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKi:  126nMAssay Description:Binding affinity against beta adrenergic receptor from rat lung tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKi:  391nMAssay Description:Binding affinity against beta adrenergic receptor from rat heart tissues was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed