Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50000808
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50397205(AR-C126532XX | AZD-6140 | AZD6140 | BRILINTA | TIC...)
Affinity DataIC50: 320nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260841(CHEMBL4077194)
Affinity DataIC50: 6.50E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260812(CHEMBL4075841)
Affinity DataIC50: 8.10E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260835(CHEMBL4065540)
Affinity DataIC50: 8.20E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260836(CHEMBL4087693)
Affinity DataIC50: 8.60E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260833(CHEMBL4079813)
Affinity DataIC50: 9.10E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260840(CHEMBL4077654)
Affinity DataIC50: 9.20E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260831(CHEMBL4075411)
Affinity DataIC50: 9.30E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260839(CHEMBL4087845)
Affinity DataIC50: 9.40E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260832(CHEMBL4067755)
Affinity DataIC50: 9.40E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260830(CHEMBL4075331)
Affinity DataIC50: 9.50E+5nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260811(CHEMBL4062156)
Affinity DataIC50: 1.32E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50234613(CHEBI:75331 | 1H-Benzo[D][1,2,3]Triazole | 1H-Benz...)
Affinity DataIC50: 7.43E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260838(CHEMBL4078992)
Affinity DataIC50: 1.07E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260837(CHEMBL4102781)
Affinity DataIC50: 1.50E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM70499(4-nitro-1H-1,2,3-benzotriazole | SMR000126045 | ML...)
Affinity DataIC50: 2.06E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260834(CHEMBL4060620)
Affinity DataIC50: 1.26E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260821(CHEMBL4093411)
Affinity DataIC50: 1.04E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260820(CHEMBL4071889)
Affinity DataIC50: 1.02E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260819(CHEMBL4076196)
Affinity DataIC50: 1.07E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260818(CHEMBL4075142)
Affinity DataIC50: 1.05E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260817(CHEMBL4100042)
Affinity DataIC50: 1.30E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260816(CHEMBL4076556)
Affinity DataIC50: 1.62E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260815(CHEMBL4084826)
Affinity DataIC50: 1.80E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260814(CHEMBL4099652)
Affinity DataIC50: 1.96E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed
TargetP2Y purinoceptor 12(Human)
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50260813(CHEMBL4073608)
Affinity DataIC50: 1.84E+6nMAssay Description:Inhibition of P2Y12 in human platelet rich plasma assessed as reduction in ADP-induced platelet aggregation pre-incubated before ADP addition and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/16/2020
Entry Details Article
PubMed