Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50001353
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50266668(CHEMBL4098545)
Affinity DataEC50:  12nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277070(CHEMBL4170976)
Affinity DataEC50:  112nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277071(CHEMBL4160365)
Affinity DataEC50:  29nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277063(CHEMBL4163731)
Affinity DataEC50:  3nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277081(CHEMBL4162383)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277073(CHEMBL4173061)
Affinity DataEC50:  0.860nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277082(CHEMBL4159003)
Affinity DataEC50:  88nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277057(CHEMBL4174154)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277074(CHEMBL4166241)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277083(CHEMBL4159426)
Affinity DataEC50:  32nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277080(CHEMBL4172444)
Affinity DataEC50:  16nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277068(CHEMBL4167169)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277056(CHEMBL4163714)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277084(CHEMBL4160347)
Affinity DataEC50:  10nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277062(CHEMBL4175452)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  7.70nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50121518(CHEMBL428139)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277081(CHEMBL4162383)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277060(CHEMBL4167331)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277053(CHEMBL4174382)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277072(CHEMBL4174404)
Affinity DataEC50:  9nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277054(CHEMBL4159275)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277082(CHEMBL4159003)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277083(CHEMBL4159426)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277084(CHEMBL4160347)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.970nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277058(CHEMBL4165144)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277069(CHEMBL4161800)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277054(CHEMBL4159275)
Affinity DataEC50:  52nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277055(CHEMBL4169653)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277056(CHEMBL4163714)
Affinity DataEC50:  0.460nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277057(CHEMBL4174154)
Affinity DataEC50:  0.860nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277058(CHEMBL4165144)
Affinity DataEC50:  3nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277059(CHEMBL4177064)
Affinity DataEC50:  2nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277055(CHEMBL4169653)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277060(CHEMBL4167331)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277061(CHEMBL4159256)
Affinity DataEC50:  0.940nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277062(CHEMBL4175452)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277063(CHEMBL4163731)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277068(CHEMBL4167169)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277053(CHEMBL4174382)
Affinity DataEC50:  5.90nMAssay Description:Agonist activity at full length human GLP1R expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277070(CHEMBL4170976)
Affinity DataEC50:  19nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277071(CHEMBL4160365)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277072(CHEMBL4174404)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277059(CHEMBL4177064)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277073(CHEMBL4173061)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277074(CHEMBL4166241)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277078(CHEMBL4170727)
Affinity DataEC50:  0.75nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277079(CHEMBL4162789)
Affinity DataEC50:  123nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277069(CHEMBL4161800)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells assessed as increase in cAMP accumulation after 20 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/28/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 53 total ) | Next | Last >>
Jump to: