Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50001125
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269734(CHEMBL4068888)
Affinity DataIC50: 45nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269737(CHEMBL4063877)
Affinity DataIC50: 48nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 50nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269742(CHEMBL4085450)
Affinity DataIC50: 79nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269741(CHEMBL4100935)
Affinity DataIC50: 89nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269744(CHEMBL4100407)
Affinity DataIC50: 145nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269743(CHEMBL4062800)
Affinity DataIC50: 170nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269740(CHEMBL4074655)
Affinity DataIC50: 200nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM67056(1-[(4-bromophenyl)methyl]-5-methylindole-2,3-dione...)
Affinity DataIC50: 204nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269735(CHEMBL4077157)
Affinity DataIC50: 229nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269749(CHEMBL4082959)
Affinity DataIC50: 263nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269750(CHEMBL4090751)
Affinity DataIC50: 398nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269733(CHEMBL4065639)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269739(CHEMBL4073582)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269736(CHEMBL4094543)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269732(CHEMBL4067881)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine as substrate by Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM14390(SILDENAFIL CITRATE | Sildenafil# | CHEMBL192 | 5-[...)
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269732(CHEMBL4067881)
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269742(CHEMBL4085450)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269736(CHEMBL4094543)
Affinity DataIC50: 9.12E+4nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269743(CHEMBL4062800)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269744(CHEMBL4100407)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269741(CHEMBL4100935)
Affinity DataIC50: 1.31E+5nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269734(CHEMBL4068888)
Affinity DataIC50: 1.58E+5nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269740(CHEMBL4074655)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269739(CHEMBL4073582)
Affinity DataIC50: 7.46E+5nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Human)
Central South University

Curated by ChEMBL
LigandPNGBDBM50269737(CHEMBL4063877)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of human PDE5A preincubated for 30 mins followed by TMB substrate addition by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/18/2020
Entry Details Article
PubMed