Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50001113
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269608(CHEMBL2407554)
Affinity DataIC50: 310nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269595(CHEMBL3911908)
Affinity DataIC50: 1.42E+3nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269607(CHEMBL4081529)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269607(CHEMBL4081529)
Affinity DataIC50: 1.78E+3nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269593(CHEMBL3964100)
Affinity DataIC50: 2.43E+3nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269594(CHEMBL3930881)
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269610(CHEMBL4067243)
Affinity DataIC50: 4.01E+3nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269595(CHEMBL3911908)
Affinity DataIC50: 4.67E+3nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells by patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269609(CHEMBL3921947)
Affinity DataIC50: 5.65E+3nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269613(CHEMBL3953555)
Affinity DataIC50: 8.78E+3nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50269611(CHEMBL3893286)
Affinity DataIC50: 1.09E+4nMAssay Description:Antagonist activity at human 5-HT6R expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP levels pre-treated for 10 mins before 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details Article
PubMed