Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002287
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456634(CHEMBL4213827)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456635(CHEMBL4213388)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456636(CHEMBL4208735)
Affinity DataEC50:  8.00E+3nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456637(CHEMBL4208460)
Affinity DataEC50:  1.60E+4nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456638(CHEMBL4205563)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456639(CHEMBL4218745)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456640(CHEMBL4214547)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456641(CHEMBL4218758)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50456642(CHEMBL4211267)
Affinity DataEC50:  6.00E+3nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Istanbul Technical University

Curated by ChEMBL
LigandPNGBDBM50159165(2S,4aR,6a(R,7R,9S,10aS,10bR)-9-(acetyloxy)-2-(fura...)
Affinity DataEC50:  0.0420nMAssay Description:Agonist activity at human kappa-type opioid receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed