Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50000667
TargetProteasome subunit beta type-5(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50257325(CHEMBL4090056)
Affinity DataKi:  375nMAssay Description:Irreversible inhibition of human 20S proteasome beta5 subunit using suc-LLVY-AMC as substrate after 4 hrs at 30 mins time interval by fluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50257327(CHEMBL4067938)
Affinity DataKi:  3.74E+3nMAssay Description:Irreversible inhibition of human 20S proteasome beta5 subunit using suc-LLVY-AMC as substrate after 4 hrs at 30 mins time interval by fluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2019
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
University of California

Curated by ChEMBL
LigandPNGBDBM50257326(CHEMBL4086345)
Affinity DataKi:  3.92E+4nMAssay Description:Irreversible inhibition of human 20S proteasome beta5 subunit using suc-LLVY-AMC as substrate after 4 hrs at 30 mins time interval by fluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2019
Entry Details Article
PubMed