Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50000584
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217112BDBM217112(US9302989, 407)
Affinity DataKi:  1nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254198BDBM50254198(CHEMBL4060799)
Affinity DataKi:  1.5nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217057BDBM217057(US9302989, 349)
Affinity DataKi:  1.60nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254199BDBM50254199(CHEMBL4083505)
Affinity DataKi:  1.70nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254216BDBM50254216(CHEMBL4096471)
Affinity DataKi:  1.90nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254215BDBM50254215(CHEMBL4089003)
Affinity DataKi:  2.5nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50435350BDBM50435350(CHEMBL17289)
Affinity DataKi:  3nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217040BDBM217040(US9302989, 332)
Affinity DataKi:  3nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81395BDBM81395(APO-866 | US20240327418, Example FK866 | US2024030...)
Affinity DataKi:  3nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254212BDBM50254212(CHEMBL4076064)
Affinity DataKi:  3.90nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254192BDBM50254192(CHEMBL4105475)
Affinity DataKi:  4.30nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215830BDBM215830(US9302989, 25)
Affinity DataKi:  4.70nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217170BDBM217170(US9302989, 608)
Affinity DataKi:  4.90nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254214BDBM50254214(CHEMBL4086819)
Affinity DataKi:  5.10nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217078BDBM217078(US9302989, 370)
Affinity DataKi:  5.40nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254184BDBM50254184(CHEMBL4082366)
Affinity DataKi:  5.60nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 216345BDBM216345(US9302989, 290)
Affinity DataKi:  7.5nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215825BDBM215825(US9302989, 20)
Affinity DataKi:  7.90nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215806BDBM215806(US9302989, 1)
Affinity DataKi:  9nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254197BDBM50254197(CHEMBL4077485)
Affinity DataKi:  9.40nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215841BDBM215841(US9302989, 36)
Affinity DataKi:  11nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215848BDBM215848(US9302989, 43)
Affinity DataKi:  13nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 216082BDBM216082(US9302989, 420)
Affinity DataKi:  13nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254187BDBM50254187(CHEMBL4062838)
Affinity DataKi:  14nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215857BDBM215857(US9302989, 53)
Affinity DataKi:  14nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217111BDBM217111(US9302989, 406)
Affinity DataKi:  15nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215863BDBM215863(US9302989, 59)
Affinity DataKi:  16nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215871BDBM215871(US9302989, 67)
Affinity DataKi:  17nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 216948BDBM216948(US9302989, 1028)
Affinity DataKi:  18nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217044BDBM217044(US9302989, 336)
Affinity DataKi:  19nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215877BDBM215877(US9302989, 73)
Affinity DataKi:  19nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 216052BDBM216052(US9302989, 252)
Affinity DataKi:  19nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254213BDBM50254213(CHEMBL4076641)
Affinity DataKi:  21nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217027BDBM217027(US9302989, 319)
Affinity DataKi:  23nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215890BDBM215890(US9302989, 86)
Affinity DataKi:  23nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 215895BDBM215895(US9302989, 91)
Affinity DataKi:  24nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217157BDBM217157(US9302989, 574)
Affinity DataKi:  57nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254189BDBM50254189(CHEMBL4077254)
Affinity DataKi:  58nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 216009BDBM216009(US9302989, 209)
Affinity DataKi:  104nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254185BDBM50254185(CHEMBL4081887)
Affinity DataKi:  112nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254186BDBM50254186(CHEMBL4099778)
Affinity DataKi:  160nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217207BDBM217207(US9302989, 808)
Affinity DataKi:  350nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50439314BDBM50439314(CHEMBL2419508)
Affinity DataKi:  487nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 216050BDBM216050(US9302989, 250)
Affinity DataKi:  560nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 253899BDBM253899(US9459250, E104)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254184BDBM50254184(CHEMBL4082366)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254191BDBM50254191(CHEMBL4090863)
Affinity DataKi: >8.90E+3nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetNicotinamide phosphoribosyltransferase(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254190BDBM50254190(CHEMBL4062656)
Affinity DataKi: >9.00E+3nMAssay Description:Inhibition of C-terminal His-tagged human recombinant NAMPT using FK866 or isoindoline urea-based Oregon green (488) probe incubated for 3 hrs by TR-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50254184BDBM50254184(CHEMBL4082366)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 217116BDBM217116(US9302989, 411)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CYP2C9 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2019
Entry Details Article
PubMed
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