Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 50049050
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233514(CHEMBL4064131)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233510(CHEMBL4095058)
Affinity DataEC50:  1.34E+3nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233517(CHEMBL4066466)
Affinity DataEC50:  313nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233496(CHEMBL4075703)
Affinity DataEC50:  680nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233495(CHEMBL4102357)
Affinity DataEC50:  1.88E+3nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233493(CHEMBL4070895)
Affinity DataEC50:  3.73E+3nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233516(CHEMBL4097990)
Affinity DataEC50:  2.51E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233492(CHEMBL4097059)
Affinity DataEC50:  1.58E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233490(CHEMBL4089352)
Affinity DataEC50:  930nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233515(CHEMBL4068168)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233488(CHEMBL4060315)
Affinity DataEC50:  310nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233487(CHEMBL4091882)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233486(CHEMBL4084125)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233485(CHEMBL4102107)
Affinity DataEC50:  4.31E+3nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233513(CHEMBL4061329)
Affinity DataEC50:  440nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233484(CHEMBL4083189)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233482(CHEMBL4072719)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233512(CHEMBL4101442)
Affinity DataEC50:  2.05E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233480(CHEMBL4102817)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233478(CHEMBL4084863)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233511(CHEMBL4064931)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233476(CHEMBL4087370)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233475(CHEMBL4065966)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233515(CHEMBL4068168)
Affinity DataEC50:  321nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233509(CHEMBL4074596)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233517(CHEMBL4066466)
Affinity DataEC50:  3.05E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233508(CHEMBL4092168)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233483(CHEMBL4099616)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233481(CHEMBL4062174)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233477(CHEMBL4092628)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233519(CHEMBL4079911)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233518(CHEMBL4104842)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233474(CHEMBL4081476)
Affinity DataEC50:  520nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233516(CHEMBL4097990)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233510(CHEMBL4095058)
Affinity DataEC50:  3.52E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233514(CHEMBL4064131)
Affinity DataEC50:  1.25E+4nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233513(CHEMBL4061329)
Affinity DataEC50:  10nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233512(CHEMBL4101442)
Affinity DataEC50:  330nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233511(CHEMBL4064931)
Affinity DataEC50:  4.81E+3nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233503(CHEMBL4095497)
Affinity DataEC50:  3.82E+4nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233519(CHEMBL4079911)
Affinity DataEC50:  2.93E+3nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233518(CHEMBL4104842)
Affinity DataEC50:  550nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233494(CHEMBL4059508)
Affinity DataEC50:  770nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233491(CHEMBL4079040)
Affinity DataEC50:  390nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233489(CHEMBL4088541)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233486(CHEMBL4084125)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Human)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233497(CHEMBL4069934)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at TGR5 in human NCI-H716 cells assessed as increase in cAMP accumulation after 40 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233496(CHEMBL4075703)
Affinity DataEC50:  300nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233495(CHEMBL4102357)
Affinity DataEC50:  120nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
TargetG-protein coupled bile acid receptor 1(Mouse)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50233494(CHEMBL4059508)
Affinity DataEC50:  50nMAssay Description:Agonist activity at TGR5 in mouse STC1 cells assessed as increase in cAMP accumulation after 40 mins by mass spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2019
Entry Details Article
PubMed
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