Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50049045
TargetE3 ubiquitin-protein ligase XIAP(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50233420(CHEMBL4092271)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of His-tagged XIAP BIR3 (241 to 356 residues) (unknown origin) using fluorescein labeled SMAC peptide as substrate after 60 mins by HTRF a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2019
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50233421(CHEMBL4075941)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of His-tagged XIAP BIR3 (241 to 356 residues) (unknown origin) using fluorescein labeled SMAC peptide as substrate after 60 mins by HTRF a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2019
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50233423(CHEMBL4091364)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of His-tagged XIAP BIR3 (241 to 356 residues) (unknown origin) using fluorescein labeled SMAC peptide as substrate after 60 mins by HTRF a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2019
Entry Details Article
PubMed
TargetE3 ubiquitin-protein ligase XIAP(Human)
Therachem Research Medilab (India)

Curated by ChEMBL
LigandPNGBDBM50233422(CHEMBL4101748)
Affinity DataIC50: 119nMAssay Description:Inhibition of His-tagged XIAP BIR3 (241 to 356 residues) (unknown origin) using fluorescein labeled SMAC peptide as substrate after 60 mins by HTRF a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/2/2019
Entry Details Article
PubMed