Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50049003
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232718(CHEMBL4096670)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232706(CHEMBL4068690 | US11046670, Table 6.2)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232702(CHEMBL4095894)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232721(CHEMBL4094368)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232722(CHEMBL4071404)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232705(CHEMBL4060037)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232701(CHEMBL4072304 | US11046670, Table 6.1)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232707(CHEMBL4062762)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232708(CHEMBL4090715)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232702(CHEMBL4095894)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232700(CHEMBL4099261)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232728(CHEMBL4074313)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232704(CHEMBL4081942)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232722(CHEMBL4071404)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232717(CHEMBL4102062)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232721(CHEMBL4094368)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232711(CHEMBL4085576)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232709(CHEMBL4098442 | US11046670, Table 6.3)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232710(CHEMBL4093176)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232719(CHEMBL4068573)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232738(CHEMBL4064084)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232749(CHEMBL4095749 | US11046670, Table 6.5)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232713(CHEMBL4077724)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232708(CHEMBL4090715)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232742(CHEMBL4065699 | US11046670, Table 6.4)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232707(CHEMBL4062762)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232700(CHEMBL4099261)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232709(CHEMBL4098442 | US11046670, Table 6.3)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232704(CHEMBL4081942)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232713(CHEMBL4077724)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232718(CHEMBL4096670)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232699(CHEMBL4091526)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232735(CHEMBL4069441 | US11046670, Compound 34)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232714(CHEMBL4101057)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232712(CHEMBL4092498 | US11046670, Compound 28)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232716(CHEMBL4072427)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232746(CHEMBL4063708 | US11046670, Compound 32)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232710(CHEMBL4093176)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232715(CHEMBL4093323)
Affinity DataKi:  108nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232715(CHEMBL4093323)
Affinity DataKi:  111nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232716(CHEMBL4072427)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232717(CHEMBL4102062)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232706(CHEMBL4068690 | US11046670, Table 6.2)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232711(CHEMBL4085576)
Affinity DataKi:  172nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232705(CHEMBL4060037)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232701(CHEMBL4072304 | US11046670, Table 6.1)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232699(CHEMBL4091526)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma intracellular receptor 2(Rat)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232714(CHEMBL4101057)
Affinity DataKi:  297nMAssay Description:Displacement of [3H]-ditolylguanidine from sigma2 receptor in rat PC12 cells in presence of (+)-pentazocine by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232749(CHEMBL4095749 | US11046670, Table 6.5)
Affinity DataKi:  413nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Guinea pig)
The University of Texas At Austin

Curated by ChEMBL
LigandPNGBDBM50232719(CHEMBL4068573)
Affinity DataKi:  473nMAssay Description:Displacement of [3H]-(+)-pentazocine from guinea pig brain sigma1 receptor by PDSP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2019
Entry Details Article
PubMed
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