Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50000509
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252033(CHEMBL4078023)
Affinity DataIC50: 20nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252035(CHEMBL4064361)
Affinity DataIC50: 20nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252089(CHEMBL4083642)
Affinity DataIC50: 40nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 60nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252090(CHEMBL4063890)
Affinity DataIC50: 60nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252091(CHEMBL4102284)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251945(CHEMBL4100075)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251946(CHEMBL4104427)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252043(CHEMBL4093642)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251947(CHEMBL4081727)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252035(CHEMBL4064361)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251948(CHEMBL4075241)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252090(CHEMBL4063890)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251949(CHEMBL4094546)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251946(CHEMBL4104427)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252033(CHEMBL4078023)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252034(CHEMBL4085902)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251948(CHEMBL4075241)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252089(CHEMBL4083642)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252091(CHEMBL4102284)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252043(CHEMBL4093642)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (unknown origin) (645 to 1186 residues) expressed in baculovirus infected Sf-9 cells pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251949(CHEMBL4094546)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251945(CHEMBL4100075)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50252034(CHEMBL4085902)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Wuhan University of Technology

Curated by ChEMBL
LigandPNGBDBM50251947(CHEMBL4081727)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of FAK (unknown origin) assembly preincubated with enzyme followed by GTP addition measured after 20 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2019
Entry Details Article
PubMed