Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50000372
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50249042(CHEMBL4087272)
Affinity DataKd:  8.50E+4nMAssay Description:Binding affinity to partial length human DNA-tagged CBP (R1081 to G1197 residues) expressed in bacterial expression system by qPCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50249043(CHEMBL4077137)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to partial length human DNA-tagged CBP (R1081 to G1197 residues) expressed in bacterial expression system by qPCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50249043(CHEMBL4077137)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of histone H4 tetraacetylated peptide binding to human CBP by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Z£Rich

Curated by ChEMBL
LigandPNGBDBM50249042(CHEMBL4087272)
Affinity DataIC50: 4.55E+5nMAssay Description:Inhibition of histone H4 tetraacetylated peptide binding to human CBP by Alphascreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)