Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50000484
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251300(CHEMBL4066684)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251300(CHEMBL4066684)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Flt-3 (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPlatelet-derived growth factor receptor beta(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251300(CHEMBL4066684)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of PDGFRbeta (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251333(CHEMBL4093275)
Affinity DataIC50: 5nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251304(CHEMBL4087981)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251311(CHEMBL4104755)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251293(CHEMBL4068286)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251324(CHEMBL4089464)
Affinity DataIC50: 10nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251303(CHEMBL4078189)
Affinity DataIC50: 10nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251332(CHEMBL4102463)
Affinity DataIC50: 11nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251312(CHEMBL4066710)
Affinity DataIC50: 12nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251337(CHEMBL4062107)
Affinity DataIC50: 13nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251299(CHEMBL4079155)
Affinity DataIC50: 14nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251294(CHEMBL4097171)
Affinity DataIC50: 15nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251302(CHEMBL4094711)
Affinity DataIC50: 18nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251326(CHEMBL4087017)
Affinity DataIC50: 18nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251313(CHEMBL4075470)
Affinity DataIC50: 18nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251309(CHEMBL4101008)
Affinity DataIC50: 19nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251325(CHEMBL4104881)
Affinity DataIC50: 20nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251301(CHEMBL4067260)
Affinity DataIC50: 22nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251322(CHEMBL4076617)
Affinity DataIC50: 29nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251291(CHEMBL4088695)
Affinity DataIC50: 32nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251334(CHEMBL4062885)
Affinity DataIC50: 34nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251310(CHEMBL4074260)
Affinity DataIC50: 35nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251315(CHEMBL4097410)
Affinity DataIC50: 36nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251335(CHEMBL4080532)
Affinity DataIC50: 40nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251317(CHEMBL4061741)
Affinity DataIC50: 41nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251305(CHEMBL4065638)
Affinity DataIC50: 41nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251306(CHEMBL4085528)
Affinity DataIC50: 42nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251316(CHEMBL4078622)
Affinity DataIC50: 45nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251292(CHEMBL4066651)
Affinity DataIC50: 46nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251308(CHEMBL4084557)
Affinity DataIC50: 47nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251323(CHEMBL4091384)
Affinity DataIC50: 49nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251307(CHEMBL4103455)
Affinity DataIC50: 56nMAssay Description:Inhibition of c-Met (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251300(CHEMBL4066684)
Affinity DataIC50: 319nMAssay Description:Inhibition of c-Kit (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251300(CHEMBL4066684)
Affinity DataIC50: 672nMAssay Description:Inhibition of VEGFR-2 (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Jiangxi Science and Technology Normal University

Curated by ChEMBL
LigandPNGBDBM50251300(CHEMBL4066684)
Affinity DataIC50: 725nMAssay Description:Inhibition of EGFR (unknown origin) using poly (Glu, Tyr) 4:1 as substrate after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2019
Entry Details Article
PubMed