BindingDB PrimarySearch

Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50000939

Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Xi'An Jiaotong University

Curated by ChEMBL

BDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)

IC50: 2.70nMAssay Description:Inhibition of PI3K p110delta/p85alpha (unknown origin) using lipid substrate after 40 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Purchase CHEMBL PC cid PC sid PDB Similars

Date in BDB:
2/10/2020
Entry Details Article
PubMed PDB

3D Structure (crystal)

Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Xi'An Jiaotong University

Curated by ChEMBL

BDBM50265448(CHEMBL4078784)

IC50: 9.30nMAssay Description:Inhibition of PI3K p110delta/p85alpha (unknown origin) using lipid substrate after 40 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid Similars

Date in BDB:
2/10/2020
Entry Details Article
PubMed

Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Human)
Xi'An Jiaotong University

Curated by ChEMBL

BDBM50265455(CHEMBL4087607)

IC50: 9.70nMAssay Description:Inhibition of PI3K p110delta/p85alpha (unknown origin) using lipid substrate after 40 mins by kinase-glo luminescence assayMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

PC cid PC sid Similars

Date in BDB:
2/10/2020
Entry Details Article
PubMed