Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50000938
TargetDeath-associated protein kinase 1(Human)
West Virginia University

Curated by ChEMBL
LigandPNGBDBM50265392(CHEMBL4088576)
Affinity DataEC50:  3.95E+4nMAssay Description:Activation of human DAPK1 using KKLNRTLSFAEPG as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
West Virginia University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.121nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details Article
PubMed
TargetDeath-associated protein kinase 1(Human)
West Virginia University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human DAPK1 using KKLNRTLSFAEPG as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details Article
PubMed
TargetERO1-like protein alpha(Mouse)
West Virginia University

Curated by ChEMBL
LigandPNGBDBM50265447(CHEMBL4060344)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of GST-SMT3-tagged mouse ERO1alpha (23 to 464 residues) expressed in Escherichia coli rosetta (DE3) using reduced thioredoxin as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
West Virginia University

Curated by ChEMBL
LigandPNGBDBM50265392(CHEMBL4088576)
Affinity DataIC50: 4.08E+3nMAssay Description:Inhibition of human PIM3 using RSRHSSYPAGT as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details Article
PubMed
TargetAlbumin(Bovine)
West Virginia University

Curated by ChEMBL
LigandPNGBDBM50265392(CHEMBL4088576)
Affinity DataIC50: 2.33E+4nMAssay Description:Binding affinity to bovine serum albumin by tryptophan quenching based HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/10/2020
Entry Details Article
PubMed