Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50049233
TargetPotassium voltage-gated channel subfamily A member 1(Human)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin) expressed in HEK293 cells by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Rat)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237249(CHEMBL4076021)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of recombinant rat Kv1.1 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Rat)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)4 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Rat)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant rat Kv1.1 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of Kv1.4 (unknown origin) expressed in HEK293 cells by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1/2(Rat)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)3/Kv1.2 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1/2(Rat)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)2/Kv(1.2)2 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM10458(pyridin-4-amine | CHEMBL284348 | 4-Aminopyridine 1...)
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50101817(CHEBI:7565 | Adalat | Adalat Cc | Afeditab Cr | BA...)
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1/2(Rat)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat Kv1.1/Kv(1.2)3 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 2(Rat)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat Kv1.2(4) expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50004704(Acetic acid 5-(2-dimethylamino-ethyl)-2-(4-methoxy...)
Affinity DataIC50: 1.44E+5nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 1(Human)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50131434(CHEMBL652 | Tambocor | N-Piperidin-2-ylmethyl-2,5-...)
Affinity DataIC50: 2.09E+5nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/3/2019
Entry Details Article
PubMed