Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50049220
Affinity DataEC50: 5nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.400nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.70nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.300nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.90nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.10nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.90nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.90nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at recombinant human kappa-type opioid receptor expressed in HEK293 cells after 30 mins by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.630nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.650nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.820nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.820nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.950nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.970nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 0.980nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]U-69,593 from kappa-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Guinea pig)
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Dr. August Wolff Gmbh & Co. Kg Arzneimittel
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]DAMGO from mu-type opioid receptor in guinea pig brain membranes after 120 mins by solid scintillation countingMore data for this Ligand-Target Pair
