Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 7849
TargetGag-Pol polyprotein(HIV-1)
Jaipur National University

LigandPNGBDBM222174(N-(2-(2,3-Dioxoindolin-1-yl)acetyl)-4,6-dimethyl-2...)
Affinity DataIC50: 64nMT: 2°CAssay Description:To a lysis buffer (20 μl), 4-6 ng recombinant HIV-1-RT was added in separate reaction tubes. Lysis buffer without HIV-1-RT was used as a negative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2017
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Jaipur National University

LigandPNGBDBM222175(N-(2-(2,3-Dioxoindolin-1-yl)acetyl)-4-ethyl-6-meth...)
Affinity DataIC50: 67nMT: 2°CAssay Description:To a lysis buffer (20 μl), 4-6 ng recombinant HIV-1-RT was added in separate reaction tubes. Lysis buffer without HIV-1-RT was used as a negative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2017
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Jaipur National University

LigandPNGBDBM222178(Rilpivirine)
Affinity DataIC50: 68nMT: 2°CAssay Description:To a lysis buffer (20 μl), 4-6 ng recombinant HIV-1-RT was added in separate reaction tubes. Lysis buffer without HIV-1-RT was used as a negative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGag-Pol polyprotein(HIV-1)
Jaipur National University

LigandPNGBDBM222176(N-(2-(2,3-Dioxoindolin-1-yl)acetyl)-6-methyl-2-oxo...)
Affinity DataIC50: 100nMT: 2°CAssay Description:To a lysis buffer (20 μl), 4-6 ng recombinant HIV-1-RT was added in separate reaction tubes. Lysis buffer without HIV-1-RT was used as a negative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2017
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Jaipur National University

LigandPNGBDBM222177(4-(4-Chlorophenyl)-N-(2-(2,3-dioxoindolin-1-yl)ace...)
Affinity DataIC50: 100nMT: 2°CAssay Description:To a lysis buffer (20 μl), 4-6 ng recombinant HIV-1-RT was added in separate reaction tubes. Lysis buffer without HIV-1-RT was used as a negative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2017
Entry Details Article
PubMed
TargetGag-Pol polyprotein(HIV-1)
Jaipur National University

LigandPNGBDBM1434(BI-RG-587 | 2-cyclopropyl-7-methyl-2,4,9,15-tetraa...)
Affinity DataIC50: 100nMT: 2°CAssay Description:To a lysis buffer (20 μl), 4-6 ng recombinant HIV-1-RT was added in separate reaction tubes. Lysis buffer without HIV-1-RT was used as a negative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2017
Entry Details Article
PubMed