Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50049027
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233221(CHEMBL4064160)
Affinity DataEC50:  5.30nMAssay Description:Inhibition of Nav1.2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233222(CHEMBL4082248)
Affinity DataEC50:  79nMAssay Description:Inhibition of Nav1.2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233224(CHEMBL4070670)
Affinity DataEC50:  120nMAssay Description:Inhibition of Nav1.2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233223(CHEMBL4060338)
Affinity DataEC50:  12nMAssay Description:Inhibition of Nav1.2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233223(CHEMBL4060338)
Affinity DataIC50: 0.280nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced tail current by whole cell patch clamp method re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233223(CHEMBL4060338)
Affinity DataIC50: 0.450nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced sustained current by whole cell patch clamp meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233224(CHEMBL4070670)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced tail current by whole cell patch clamp method re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233224(CHEMBL4070670)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced sustained current by whole cell patch clamp meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233222(CHEMBL4082248)
Affinity DataIC50: 7.5nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced sustained current by whole cell patch clamp meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233221(CHEMBL4064160)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced sustained current by whole cell patch clamp meth...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233222(CHEMBL4082248)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced tail current by whole cell patch clamp method re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed
TargetSodium channel protein type 2 subunit alpha(Human)
Tohoku University

Curated by ChEMBL
LigandPNGBDBM50233221(CHEMBL4064160)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at human Nav1.2 expressed in HEK293T cells assessed as inhibition of VTD-induced tail current by whole cell patch clamp method re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2019
Entry Details Article
PubMed