Compile Data Set for Download or QSAR
Report error Found 66 Enz. Inhib. hit(s) with all data for entry = 50048948
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230956(CHEMBL4079784)
Affinity DataEC50:  0.700nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230961(CHEMBL4062947)
Affinity DataEC50:  9.5nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230960(CHEMBL4089965)
Affinity DataEC50: >1.00E+3nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230955(CHEMBL4102177)
Affinity DataEC50:  0.200nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataEC50:  1.40nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230952(CHEMBL4079699)
Affinity DataEC50:  1.10nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230961(CHEMBL4062947)
Affinity DataEC50:  0.200nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230959(CHEMBL4084612)
Affinity DataEC50:  0.0900nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230958(CHEMBL4071572)
Affinity DataEC50:  0.200nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230960(CHEMBL4089965)
Affinity DataEC50:  0.800nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataEC50:  0.180nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230952(CHEMBL4079699)
Affinity DataEC50:  31nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230951(CHEMBL4095210)
Affinity DataEC50:  90nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230959(CHEMBL4084612)
Affinity DataEC50:  19nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230958(CHEMBL4071572)
Affinity DataEC50:  1.62E+3nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230957(CHEMBL4082097)
Affinity DataEC50: >1.00E+3nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230956(CHEMBL4079784)
Affinity DataEC50:  65nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230955(CHEMBL4102177)
Affinity DataEC50:  0.800nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230957(CHEMBL4082097)
Affinity DataEC50:  0.400nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230951(CHEMBL4095210)
Affinity DataEC50:  0.100nMAssay Description:Intrinsic activity at human MT2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230960(CHEMBL4089965)
Affinity DataKi:  0.0300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230959(CHEMBL4084612)
Affinity DataKi:  0.0900nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230961(CHEMBL4062947)
Affinity DataKi:  0.0900nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230951(CHEMBL4095210)
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.100nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.120nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230955(CHEMBL4102177)
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230958(CHEMBL4071572)
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230955(CHEMBL4102177)
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230957(CHEMBL4082097)
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230965(CHEMBL4061905)
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230956(CHEMBL4079784)
Affinity DataKi:  0.300nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.310nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230952(CHEMBL4079699)
Affinity DataKi:  0.400nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230969(CHEMBL4070527)
Affinity DataKi:  0.5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230959(CHEMBL4084612)
Affinity DataKi:  0.600nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230961(CHEMBL4062947)
Affinity DataKi:  0.800nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230966(CHEMBL4100108)
Affinity DataKi:  1nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230951(CHEMBL4095210)
Affinity DataKi:  2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230958(CHEMBL4071572)
Affinity DataKi:  2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230952(CHEMBL4079699)
Affinity DataKi:  4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230962(CHEMBL4094436)
Affinity DataKi:  4nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230960(CHEMBL4089965)
Affinity DataKi:  5nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230964(CHEMBL4097693)
Affinity DataKi:  6nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230957(CHEMBL4082097)
Affinity DataKi:  7nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230956(CHEMBL4079784)
Affinity DataKi:  8nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230966(CHEMBL4100108)
Affinity DataKi:  16nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230965(CHEMBL4061905)
Affinity DataKi:  19nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
Universities of Lille

Curated by ChEMBL
LigandPNGBDBM50230971(CHEMBL4073867)
Affinity DataKi:  22nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in HEK or CHO cell membranes after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2019
Entry Details Article
PubMed
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