Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50048987
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232473(CHEMBL4087627)
Affinity DataIC50: 202nMAssay Description:Inhibition of human liver cathepsin-L using Z-FR-AMC as substrate preincubated for 5 mins followed by substrate addition measured at 15 sec interval ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232474(CHEMBL4066272)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-L using Z-FR-AMC as substrate preincubated for 5 mins followed by substrate addition measured at 15 sec interval ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232475(CHEMBL4091924)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-L using Z-FR-AMC as substrate preincubated for 5 mins followed by substrate addition measured at 15 sec interval ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232476(CHEMBL4071100)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-L using Z-FR-AMC as substrate preincubated for 5 mins followed by substrate addition measured at 15 sec interval ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232477(CHEMBL4074889)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-B using Z-RR-AMC as substrate preincubated for 5 mins followed by substrate addition measured for 5 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232473(CHEMBL4087627)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-B using Z-RR-AMC as substrate preincubated for 5 mins followed by substrate addition measured for 5 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232479(CHEMBL4079753)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-B using Z-RR-AMC as substrate preincubated for 5 mins followed by substrate addition measured for 5 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232480(CHEMBL4104018)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-B using Z-RR-AMC as substrate preincubated for 5 mins followed by substrate addition measured for 5 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232477(CHEMBL4074889)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-L using Z-FR-AMC as substrate preincubated for 5 mins followed by substrate addition measured at 15 sec interval ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232474(CHEMBL4066272)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-B using Z-RR-AMC as substrate preincubated for 5 mins followed by substrate addition measured for 5 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232475(CHEMBL4091924)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin-B using Z-RR-AMC as substrate preincubated for 5 mins followed by substrate addition measured for 5 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330030([(3-Bromophenyl)-(3-hydroxyphenyl)-ketone]thiosemi...)
Affinity DataKi:  3.70nMAssay Description:Covalent/reversible inhibition of human liver cathepsin-L using Z-FR-AMC as substrate preincubated for 5 mins followed by substrate addition measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50232473(CHEMBL4087627)
Affinity DataKi:  8.40nMAssay Description:Covalent/reversible inhibition of human liver cathepsin-L using Z-FR-AMC as substrate preincubated for 5 mins followed by substrate addition measured...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details Article
PubMed