Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50049138
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50153300(1-[2-Chloro-6-(3,4,5-trihydroxy-6-hydroxymethyl-te...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235128(CHEMBL4082151)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235138(CHEMBL4082869)
Affinity DataIC50: 12nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235139(CHEMBL4063790)
Affinity DataIC50: 18nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235127(CHEMBL1645378)
Affinity DataIC50: 20nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235126(CHEMBL4091589)
Affinity DataIC50: 21nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235125(CHEMBL4072377)
Affinity DataIC50: 22nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235124(CHEMBL4099324)
Affinity DataIC50: 23nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM20875(CHEMBL245067 | JMC511145 Compound 1 | 1-(2,4-dihyd...)
Affinity DataIC50: 67nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM20875(CHEMBL245067 | JMC511145 Compound 1 | 1-(2,4-dihyd...)
Affinity DataIC50: 499nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50153300(1-[2-Chloro-6-(3,4,5-trihydroxy-6-hydroxymethyl-te...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM93618(3-phenyl-1-[2,4,6-tris(oxidanyl)phenyl]propan-1-on...)
Affinity DataIC50: 7.90E+3nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235132(CHEMBL4092575)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235128(CHEMBL4082151)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235140(CHEMBL4084816)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235127(CHEMBL1645378)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235136(CHEMBL2234026)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235139(CHEMBL4063790)
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235129(CHEMBL4068024)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM23446(3-(4-hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop...)
Affinity DataIC50: 1.24E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235131(CHEMBL4101262)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235126(CHEMBL4091589)
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235125(CHEMBL4072377)
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM93618(3-phenyl-1-[2,4,6-tris(oxidanyl)phenyl]propan-1-on...)
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235130(CHEMBL4074544)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235124(CHEMBL4099324)
Affinity DataIC50: 1.56E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235132(CHEMBL4092575)
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235129(CHEMBL4068024)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235130(CHEMBL4074544)
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235140(CHEMBL4084816)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235135(4-METHOXYL-2',4',6'-TRIHYDROXYCHALCONE)
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM23446(3-(4-hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop...)
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235131(CHEMBL4101262)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235138(CHEMBL4082869)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235133(CHEMBL4071789)
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235137(4-BROMO-2',4',6'-TRIHYDROXYCHALCONE)
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50042976(2',4',6'-trihydroxychalcone | (E)-3-phenyl-1-(2,4,...)
Affinity DataIC50: 2.54E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235123(4-FLUORO-2',4',6'-TRIHYDROXYCHALCONE)
Affinity DataIC50: 2.56E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235134(CHEMBL4082294)
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235141(CHEMBL4100313)
Affinity DataIC50: 2.62E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235141(CHEMBL4100313)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50042976(2',4',6'-trihydroxychalcone | (E)-3-phenyl-1-(2,4,...)
Affinity DataIC50: 3.33E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235134(CHEMBL4082294)
Affinity DataIC50: 3.39E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235136(CHEMBL2234026)
Affinity DataIC50: 3.41E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235137(4-BROMO-2',4',6'-TRIHYDROXYCHALCONE)
Affinity DataIC50: 3.46E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235135(4-METHOXYL-2',4',6'-TRIHYDROXYCHALCONE)
Affinity DataIC50: 5.09E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 2(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235123(4-FLUORO-2',4',6'-TRIHYDROXYCHALCONE)
Affinity DataIC50: 5.17E+4nMAssay Description:Inhibition of human SGLT2 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Human)
Universidade De Lisboa

Curated by ChEMBL
LigandPNGBDBM50235133(CHEMBL4071789)
Affinity DataIC50: 5.26E+4nMAssay Description:Inhibition of human SGLT1 expressed in HEK293 cells assessed as reduction in 2-deoxyglucose uptake pretreated for 10 mins followed by 2-deoxyglucose ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2019
Entry Details Article
PubMed