Report error Found 118 Enz. Inhib. hit(s) with all data for entry = 50048942
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 101nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 116nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 117nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 125nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 182nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 213nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 226nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 241nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 292nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 329nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 395nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 441nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 534nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 603nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 686nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 2.04E+3nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 2.64E+3nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataIC50: 2.67E+3nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 5.70nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Mouse)
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
National Institute On Alcohol Abuse and Alcoholism
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]CP55940 from mouse brain CB1R expressed in CHOK1 cell membranesMore data for this Ligand-Target Pair
