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Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50000989
TargetBromodomain-containing protein 9(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataKd:  1.13E+3nMAssay Description:Binding affinity to human BRD9 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain and PHD finger-containing protein 3(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataKd:  940nMAssay Description:Binding affinity to human BRPF3 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataKd:  210nMAssay Description:Binding affinity to human BRPF2 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataKd:  40nMAssay Description:Binding affinity to human BRPF1 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249785(CHEMBL4069814)
Affinity DataIC50: 9nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267002(CHEMBL4097011)
Affinity DataIC50: 15nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249770(CHEMBL4076056)
Affinity DataIC50: 43nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267005(CHEMBL4099455)
Affinity DataIC50: 44nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 48nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249816(CHEMBL4103432)
Affinity DataIC50: 56nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267004(CHEMBL4096095)
Affinity DataIC50: 60nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267003(CHEMBL4081438)
Affinity DataIC50: 62nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249772(CHEMBL4067436)
Affinity DataIC50: 65nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 7(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 82nMAssay Description:Inhibition of human BRD7 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249785(CHEMBL4069814)
Affinity DataIC50: 130nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 140nMAssay Description:Inhibition of human His tagged BRPF1 incubated for 30 mins followed by addition of biotinylated peptide and further incubation for 30 mins measured b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249809(CHEMBL4080511)
Affinity DataIC50: 180nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267006(CHEMBL4079041)
Affinity DataIC50: 190nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249770(CHEMBL4076056)
Affinity DataIC50: 200nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249772(CHEMBL4067436)
Affinity DataIC50: 220nMAssay Description:Inhibition of human BRD9 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267008(CHEMBL4078047)
Affinity DataIC50: 220nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267005(CHEMBL4099455)
Affinity DataIC50: 230nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain and PHD finger-containing protein 3(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 260nMAssay Description:Inhibition of human BRPF3 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249816(CHEMBL4103432)
Affinity DataIC50: 270nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 310nMAssay Description:Inhibition of human BRD9 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267008(CHEMBL4078047)
Affinity DataIC50: 420nMAssay Description:Inhibition of human BRD9 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249771(CHEMBL4070377)
Affinity DataIC50: 430nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267003(CHEMBL4081438)
Affinity DataIC50: 450nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249785(CHEMBL4069814)
Affinity DataIC50: 600nMAssay Description:Inhibition of human BRD4-BD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 760nMAssay Description:Inhibition of human His tagged BRPF2 incubated for 30 mins followed by addition of biotinylated peptide and further incubation for 30 mins measured b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267004(CHEMBL4096095)
Affinity DataIC50: 890nMAssay Description:Inhibition of human BRD9 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249770(CHEMBL4076056)
Affinity DataIC50: 910nMAssay Description:Inhibition of human BRD9 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain and PHD finger-containing protein 3(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249770(CHEMBL4076056)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human BRPF3 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human His tagged BRD9 incubated for 30 mins followed by addition of biotinylated peptide and further incubation for 30 mins measured by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249772(CHEMBL4067436)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249771(CHEMBL4070377)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249772(CHEMBL4067436)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human BRD4-BD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267004(CHEMBL4096095)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain and PHD finger-containing protein 3(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human His tagged BRPF3 incubated for 30 mins followed by addition of biotinylated peptide and further incubation for 30 mins measured b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267007(CHEMBL4095549)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain and PHD finger-containing protein 3(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267003(CHEMBL4081438)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human BRPF3 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 9(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267003(CHEMBL4081438)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human BRD9 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 1(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267008(CHEMBL4078047)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human BRPF2-BRD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249770(CHEMBL4076056)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human BRD4-BD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249810(CHEMBL4102050)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human BRD4-BD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267008(CHEMBL4078047)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human BRD4-BD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50157646(CHEMBL216146)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human BRPF1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50267003(CHEMBL4081438)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human BRD4-BD1 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
TargetBromodomain and PHD finger-containing protein 3(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50249772(CHEMBL4067436)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human BRPF3 expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2020
Entry Details Article
PubMed
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