Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50001147
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209759(CHEMBL3884839)
Affinity DataIC50: 0.540nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209748(CHEMBL3884960)
Affinity DataIC50: 0.630nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209760(CHEMBL3885421)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209759(CHEMBL3884839)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209653(CHEMBL3884616)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209662(CHEMBL3884569)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209657(CHEMBL3884229)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209660(CHEMBL3884281)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209748(CHEMBL3884960)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50042034(CHEMBL1077979 | CHEBI:67559 | (5Z)-7-Oxozeaenol | ...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209753(CHEMBL3884642)
Affinity DataIC50: 7nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209758(CHEMBL3884143)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50269620(CHEMBL4128584)
Affinity DataIC50: 25nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50269622(CHEMBL4129274)
Affinity DataIC50: 33nMAssay Description:Inhibition of TAK1 (unknown origin) after 60 mins by biochemical assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209651(CHEMBL3883384 | US12365664, Compound SM1-71)
Affinity DataIC50: 50nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209755(CHEMBL3884914)
Affinity DataIC50: 57nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209673(CHEMBL3883761)
Affinity DataIC50: 75nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209757(CHEMBL3884813)
Affinity DataIC50: 83nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209752(CHEMBL3885038)
Affinity DataIC50: 92nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209652(CHEMBL3884555)
Affinity DataIC50: 950nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50269616(CHEMBL4127488)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209754(CHEMBL3884293)
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50269621(CHEMBL4129949)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209756(CHEMBL3884215)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209655(CHEMBL3885053)
Affinity DataIC50: 3.01E+3nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Dana-Farber Cancer Institute

Curated by ChEMBL
LigandPNGBDBM50209654(CHEMBL3884614)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TAK1 (unknown origin) by LanthaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2020
Entry Details Article
PubMed