Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50047988
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50168000(benzo[d]oxazol-2(3H)-one | benzoxazolinone | 3H-Be...)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200114(CHEMBL3920498)
Affinity DataIC50: 6.67E+4nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200110(CHEMBL3890166)
Affinity DataIC50: 7.17E+4nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200112(CHEMBL3895218)
Affinity DataIC50: 8.93E+4nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200119(CHEMBL3896658)
Affinity DataIC50: 9.12E+4nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200111(CHEMBL3981566)
Affinity DataIC50: 1.39E+5nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetPolypeptide N-acetylgalactosaminyltransferase 2(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200111(CHEMBL3981566)
Affinity DataIC50: 4.30E+5nMAssay Description:Inhibition of ppGalNAcT2 (unknown origin) in presence of OGT, EA2 and UDP-GlcNAc incubated for 25 mins at 37 degCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetPolypeptide N-acetylgalactosaminyltransferase 2(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200114(CHEMBL3920498)
Affinity DataIC50: 6.96E+5nMAssay Description:Inhibition of ppGalNAcT2 (unknown origin) in presence of OGT, EA2 and UDP-GlcNAc incubated for 25 mins at 37 degCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200117(CHEMBL3969655)
Affinity DataIC50: 8.65E+5nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50027783(2-Ethynyl Naphtalene | CHEMBL1743361)
Affinity DataIC50: 4.00E+6nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200118(CHEMBL3924189)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50027776(4-Ethynyl Biphenyl | 4-Ethynyl-Biphenyl | CHEMBL37...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200116(CHEMBL3933877)
Affinity DataIC50: 1.96E+6nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200115(CHEMBL3892504)
Affinity DataIC50: 4.00E+6nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200113(CHEMBL3949890)
Affinity DataIC50: 3.97E+6nMAssay Description:Inhibition of OGT (unknown origin) assessed as reduction in GlcNAc transfer to CKII peptide incubated for 60 mins by HPLC methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200114(CHEMBL3920498)
Affinity DataKi:  2.86E+4nMAssay Description:Noncompetitive inhibition of OGT (unknown origin) using variable UDP-GlcNAc levels and fixed CKII peptide level by UDP-Glo glycosyltransferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200114(CHEMBL3920498)
Affinity DataKi:  5.98E+4nMAssay Description:Noncompetitive inhibition of OGT (unknown origin) using fixed UDP-GlcNAc levels and variable CKII peptide level by UDP-Glo glycosyltransferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200111(CHEMBL3981566)
Affinity DataKi:  9.20E+4nMAssay Description:Noncompetitive inhibition of OGT (unknown origin) using variable UDP-GlcNAc levels and fixed CKII peptide level by UDP-Glo glycosyltransferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed
TargetUDP-N-acetylglucosamine--peptide N-acetylglucosaminyltransferase 110 kDa subunit(Human)
University of Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50200111(CHEMBL3981566)
Affinity DataKi:  3.10E+5nMAssay Description:Noncompetitive inhibition of OGT (unknown origin) using fixed UDP-GlcNAc levels and variable CKII peptide level by UDP-Glo glycosyltransferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2018
Entry Details Article
PubMed